DE602004031163D1 - Phenylcarboxamidverbindungen zur Schmerzbehandlung - Google Patents

Phenylcarboxamidverbindungen zur Schmerzbehandlung

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Publication number
DE602004031163D1
DE602004031163D1 DE602004031163T DE602004031163T DE602004031163D1 DE 602004031163 D1 DE602004031163 D1 DE 602004031163D1 DE 602004031163 T DE602004031163 T DE 602004031163T DE 602004031163 T DE602004031163 T DE 602004031163T DE 602004031163 D1 DE602004031163 D1 DE 602004031163D1
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Germany
Prior art keywords
pain treatment
phenylene compound
compounds
animal
effective amount
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DE602004031163T
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English (en)
Inventor
Qun Sun
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Euro Celtique SA
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Euro Celtique SA
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Publication date
Application filed by Euro Celtique SA filed Critical Euro Celtique SA
Publication of DE602004031163D1 publication Critical patent/DE602004031163D1/de
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/54Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/56Amides
DE602004031163T 2003-09-22 2004-09-21 Phenylcarboxamidverbindungen zur Schmerzbehandlung Active DE602004031163D1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US50467903P 2003-09-22 2003-09-22

Publications (1)

Publication Number Publication Date
DE602004031163D1 true DE602004031163D1 (de) 2011-03-03

Family

ID=34392933

Family Applications (2)

Application Number Title Priority Date Filing Date
DE602004031163T Active DE602004031163D1 (de) 2003-09-22 2004-09-21 Phenylcarboxamidverbindungen zur Schmerzbehandlung
DE602004014791T Active DE602004014791D1 (de) 2003-09-22 2004-09-21 Zur behandlung von schmerzen geeignete phenylcarbonsäureamidverbindungen

Family Applications After (1)

Application Number Title Priority Date Filing Date
DE602004014791T Active DE602004014791D1 (de) 2003-09-22 2004-09-21 Zur behandlung von schmerzen geeignete phenylcarbonsäureamidverbindungen

Country Status (17)

Country Link
US (3) US7799807B2 (de)
EP (2) EP1664041B1 (de)
JP (2) JP4634385B2 (de)
CN (1) CN1856489A (de)
AT (2) ATE496048T1 (de)
AU (1) AU2004276251B2 (de)
CA (1) CA2537010A1 (de)
CY (2) CY1108367T1 (de)
DE (2) DE602004031163D1 (de)
DK (2) DK1664041T3 (de)
ES (2) ES2360152T3 (de)
HK (1) HK1094191A1 (de)
HR (2) HRP20080492T3 (de)
PL (2) PL1664041T3 (de)
PT (2) PT1664041E (de)
SI (2) SI1664041T1 (de)
WO (1) WO2005030766A1 (de)

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DK1664041T3 (da) 2003-09-22 2008-10-27 Euro Celtique Sa Phenylcarboxamidforbindelser, der er egnede til behandling af smerter
ATE412646T1 (de) * 2003-09-22 2008-11-15 Euro Celtique Sa Zur behandlung von schmerzen geeignete therapeutische mittel
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WO2011162409A1 (en) 2010-06-22 2011-12-29 Shionogi & Co., Ltd. Compounds having trpv1 antagonistic activity and uses thereof
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PT2723732T (pt) 2011-06-22 2017-02-17 Purdue Pharma Lp Antagonistas de trpv1 incluindo substituinte di-hidroxilo e suas utilizações
US9394293B2 (en) * 2011-08-10 2016-07-19 Purdue Pharma L.P. TRPV1 antagonists including dihydroxy substituent and uses thereof
RU2595857C2 (ru) * 2012-05-31 2016-08-27 Кинки Юниверсити Средство для профилактического и/или терапевтического лечения периферической нейропатической боли, вызываемой противораковым средством
CA2937365C (en) 2016-03-29 2018-09-18 F. Hoffmann-La Roche Ag Granulate formulation of 5-methyl-1-phenyl-2-(1h)-pyridone and method of making the same
GB201709459D0 (en) * 2017-06-14 2017-07-26 Intrabio Ltd Treatment for migraine
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