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FIG. 2 5-point Dose Response with Human PCSK9 Leads in HEK-293 Cells Treated for 24 Hr

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160 4 120

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Ribogreen Nonnalized Perecnt UTC

PCSK9 mRNA levels in Cynomolgus Monkey Primary Hepatocytes 24 Hr After ASO

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FIG. 3

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62 J0 s was no: ‘M 1181‘ luawd ‘Sn

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Plasma LDL-C at 6 wk

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g 60- vs saline m . E 40'200s§ 6° 08 6° 9 935 - q>'$ ‘$6 <3 1» 91 *9’ 9? 9.9 B Liver TG at 6 wk 60. *p=002 5°‘ vs saline 40~ . ga 30- V U) 'E 20.. 100- ‘\ ,;9°” 6° 0“ 6° 9Qqql Q;~?° Q;$’ 9» 01 01 '2?’ ‘£9 '2?’

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